Changes in tissue gadolinium biodistribution measured in an animal model exposed to four chelating agents

Jpn J Radiol. 2019 Jun;37(6):458-465. doi: 10.1007/s11604-019-00835-1. Epub 2019 Mar 30.

Abstract

Purpose: This study investigated the potential to reduce gadolinium levels in rodents after repetitive IV Gadodiamide administration using several chelating agents.

Materials and methods: The following six groups of rats were studied. Group 1: Control; Group 2: Gadodiamide only; Group 3: Meso-2,3-Dimercaptosuccinic acid (DMSA) + Gadodiamide; Group 4: N-Acetyl-L-cysteine (NAC) + Gadodiamide; Group 5: Coriandrum sativum extract + Gadodiamide; and Group 6: Deferoxamine + Gadodiamide. Brain, kidney, and blood samples were evaluated via inductively coupled plasma mass spectrometry. The brain was also evaluated histologically.

Results: Kidney gadolinium levels in Groups 4 and 5 were approximately double that of Group 2 (p = 0.033 for each). There was almost no calcification in rat hippocampus for Group 4 rodents when compared with Groups 2, 3, 5 and 6.

Conclusion: Our preliminary study shows that excretion to the kidney has a higher propensity in NAC and Coriandrum sativum groups. It may be possible to change the distribution of gadolinium by administrating several agents. NAC may lower Gadodiamide-induced mineralization in rat hippocampus.

Keywords: Coriandrum sativum; Deferoxamine; Dimercaptosuccinic acid; Gadolinium deposition; N-Acetyl-L-cysteine.

MeSH terms

  • Animals
  • Brain / metabolism
  • Chelating Agents / administration & dosage
  • Chelating Agents / pharmacokinetics*
  • Contrast Media / administration & dosage
  • Contrast Media / pharmacokinetics*
  • Cysteine / administration & dosage
  • Cysteine / blood
  • Cysteine / pharmacokinetics
  • Gadolinium / administration & dosage
  • Gadolinium / blood
  • Gadolinium / pharmacokinetics*
  • Gadolinium DTPA / administration & dosage
  • Gadolinium DTPA / blood
  • Gadolinium DTPA / pharmacokinetics
  • Kidney / metabolism
  • Male
  • Mice
  • Models, Animal
  • Rats
  • Rats, Wistar
  • Spectrophotometry, Atomic
  • Succimer / administration & dosage
  • Succimer / pharmacokinetics
  • Tissue Distribution

Substances

  • Chelating Agents
  • Contrast Media
  • gadodiamide
  • Gadolinium
  • Succimer
  • Gadolinium DTPA
  • Cysteine