The short-chain fatty acid pentanoate suppresses autoimmunity by modulating the metabolic-epigenetic crosstalk in lymphocytes

Nat Commun. 2019 Feb 15;10(1):760. doi: 10.1038/s41467-019-08711-2.

Abstract

Short-chain fatty acids (SCFAs) have immunomodulatory effects, but the underlying mechanisms are not well understood. Here we show that pentanoate, a physiologically abundant SCFA, is a potent regulator of immunometabolism. Pentanoate induces IL-10 production in lymphocytes by reprogramming their metabolic activity towards elevated glucose oxidation. Mechanistically, this reprogramming is mediated by supplying additional pentanoate-originated acetyl-CoA for histone acetyltransferases, and by pentanoate-triggered enhancement of mTOR activity. In experimental mouse models of colitis and multiple sclerosis, pentanoate-induced regulatory B cells mediate protection from autoimmune pathology. Additionally, pentanoate shows a potent histone deacetylase-inhibitory activity in CD4+ T cells, thereby reducing their IL-17A production. In germ-free mice mono-colonized with segmented filamentous bacteria (SFB), pentanoate inhibits the generation of small-intestinal Th17 cells and ameliorates SFB-promoted inflammation in the central nervous system. Taken together, by enhancing IL-10 production and suppressing Th17 cells, the SCFA pentanoate might be of therapeutic relevance for inflammatory and autoimmune diseases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Autoimmunity / drug effects*
  • CD4-Positive T-Lymphocytes / drug effects
  • CD4-Positive T-Lymphocytes / metabolism
  • Colitis / drug therapy
  • Colitis / metabolism
  • Epigenesis, Genetic / drug effects*
  • Epigenesis, Genetic / genetics*
  • Fatty Acids, Volatile / physiology
  • Fatty Acids, Volatile / therapeutic use
  • Interleukin-10 / metabolism
  • Lymphocytes / drug effects*
  • Lymphocytes / metabolism*
  • Mice
  • Multiple Sclerosis / drug therapy
  • Multiple Sclerosis / metabolism
  • Th17 Cells / drug effects
  • Th17 Cells / metabolism
  • Valerates / pharmacology*
  • Valerates / therapeutic use

Substances

  • Fatty Acids, Volatile
  • Valerates
  • Interleukin-10