Two new steroidal saponins from Maianthemum henryi and their cytotoxic activity against human HepG2 tumor cells

Nat Prod Res. 2019 Dec;33(24):3551-3558. doi: 10.1080/14786419.2018.1514605. Epub 2018 Dec 23.

Abstract

Two new steroidal saponins (1 and 2), along with four known ones (36) were obtained from the roots and rhizomes of Maianthemum henryi, their structures were determined to be spirost-5, 25(27)-diene-lβ, 3β-diol 1-O-α-L-rhamnopyranosyl-(1 → 2)-4-O-acetyl-β-D-fucopyranoside (1), (23S, 24S)-spirost-5, 25(27)-diene-lβ, 3β, 23, 24-tetrol 1-O-α-L-rhamnopyranosyl-(1 → 2)-4-O-acetyl-β-D-fucopyranoside (2), spirost-5, 25(27)-diene-lβ, 3β-diol 1-O-α-L-rhamnopyranosyl-(1 → 2)-β-D-fucopyranoside (3), spirost-5, 25(27)-diene-lβ, 3β-diol 1-O-α-L-rhamnopyranosyl-(1 → 2)-β-D-xylopyranoside (4), Henryioside A (5)、Henryioside B (6), by physicochemical properties and spectroscopic methods. In addition, their cytotoxic activity against human HepG2 tumor cells was evaluated by MTT method and all of the compounds exhibited cytotoxicity with the cells.

Keywords: Maianthemum henryi; cytotoxicity; steroidal saponins; structure evaluation.

MeSH terms

  • Antineoplastic Agents / analysis
  • Antineoplastic Agents / isolation & purification*
  • Cytotoxins / isolation & purification
  • Cytotoxins / pharmacology
  • Hep G2 Cells
  • Humans
  • Maianthemum / chemistry*
  • Molecular Structure
  • Plant Extracts / chemistry
  • Plant Extracts / therapeutic use
  • Saponins / chemistry*
  • Saponins / isolation & purification
  • Steroids / chemistry*
  • Steroids / isolation & purification

Substances

  • Antineoplastic Agents
  • Cytotoxins
  • Plant Extracts
  • Saponins
  • Steroids