Two new monoterpenoid indole alkaloids from Tabernaemontana divaricata

Nat Prod Res. 2019 Aug;33(15):2139-2144. doi: 10.1080/14786419.2018.1488707. Epub 2018 Nov 16.

Abstract

Two new monoterpenoid indole alkaloids, tabervarines A (1) and B (2), along with seven known monoterpenoid indole alkaloids, were isolated from the methanol extract of the twigs and leaves of Tabernaemontana divaricata. The structures including the absolute configurations of the new alkaloids were elucidated based on MS, NMR, and ECD calculation. The in vitro cytotoxic activities of the isolated alkaloids against several human cancer cell lines were also evaluated.

Keywords: Tabernaemontana divaricata; monoterpenoid indole alkaloids; tabervarine A; tabervarine B.

MeSH terms

  • Cell Line, Tumor
  • Drug Screening Assays, Antitumor
  • Humans
  • Molecular Structure
  • Plant Leaves / chemistry
  • Secologanin Tryptamine Alkaloids / chemistry*
  • Secologanin Tryptamine Alkaloids / isolation & purification*
  • Secologanin Tryptamine Alkaloids / pharmacology
  • Spectrum Analysis / methods
  • Tabernaemontana / chemistry*

Substances

  • Secologanin Tryptamine Alkaloids