Losartan treatment significantly attenuates the fibrotic changes in the corpus cavernosum of castrated rats

Rev Int Androl. 2020 Jan-Mar;18(1):14-20. doi: 10.1016/j.androl.2018.07.001. Epub 2018 Sep 21.

Abstract

Introduction and objectives: The aim of this study is to evaluate the effects of castration and subsequent losartan administration on the fibrosis-related parameters in the corpora cavernosa of castrated rats.

Material and methods: Twenty-four male rats were divided into four equal groups. Group 1:sham surgery plus vehicle (0.9% NaCl) (control:con), group 2:sham surgery plus losartan (con+los), group 3: castration plus vehicle (castration:cast) and group 4:castration plus losartan (cast+los). After four weeks of oral losartan treatment, corporal levels of transforming growth factor-beta (TGF-β), thrombospondin-1 (TSP-1), alpha-actin, beta-actin and fibronectin were investigated by ELISA kits. Changes in the collagen and smooth muscle content were evaluated by histological analysis with Masson trichrome staining.

Results: Initial and post-treatment body weights of rats were similar among groups. Castration significantly increased the expression of TGF-β, TSP-1 and fibronectin and resulted in a significant decrease in alpha-actin levels in the corpora cavernosa. Administration of losartan reduced the levels of TGF-β, TSP-1 and fibronectin in castrated rats. Alpha actin levels also increased after losartan treatment. Beta-actin levels were not significantly different among 4 groups. The levels of all markers were similar in group 1 and 2. Rate of fibrosis was significantly higher in castrated rats and treatment with losartan reduced this rate.

Conclusion: Castration increased the expression of fibrosis-related markers in the corpora cavernosa of rats. Administration of losartan significantly attenuated those changes and exerted an antifibrotic effect.

Keywords: Castración; Castration; Corporal fibrosis; Disfunción eréctil; Erectile dysfunction; Fibrosis corporal; Losartan; Losartán.

MeSH terms

  • Actins / analysis
  • Angiotensin II Type 1 Receptor Blockers / pharmacology*
  • Animals
  • Biomarkers / analysis
  • Body Weight
  • Collagen / analysis
  • Fibronectins / analysis
  • Fibrosis
  • Losartan / pharmacology*
  • Male
  • Muscle, Smooth / anatomy & histology
  • Orchiectomy*
  • Penis / chemistry
  • Penis / drug effects*
  • Penis / pathology
  • Rats
  • Rats, Wistar
  • Testosterone / blood
  • Thrombospondin 1 / analysis
  • Transforming Growth Factor beta / analysis

Substances

  • Actins
  • Angiotensin II Type 1 Receptor Blockers
  • Biomarkers
  • Fibronectins
  • Thrombospondin 1
  • Transforming Growth Factor beta
  • thrombospondin 1, rat
  • Testosterone
  • Collagen
  • Losartan