Studies on the conformation, enzymatic degradation, pharmacological potency, and binding properties in brain tissue of cholecystokinin-8 and new related peptides

Ann N Y Acad Sci. 1985:448:61-75. doi: 10.1111/j.1749-6632.1985.tb29907.x.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Brain / metabolism*
  • Cerebral Cortex / metabolism
  • Endopeptidases / pharmacology
  • Fluorescence
  • Humans
  • Magnetic Resonance Spectroscopy
  • Mice
  • Neprilysin
  • Protein Conformation
  • Rats
  • Receptors, Cell Surface / drug effects
  • Receptors, Cholecystokinin
  • Sincalide / analysis
  • Sincalide / metabolism*
  • Sincalide / pharmacology
  • Structure-Activity Relationship
  • Swine
  • Synaptosomes / metabolism

Substances

  • Receptors, Cell Surface
  • Receptors, Cholecystokinin
  • Endopeptidases
  • Neprilysin
  • Sincalide