Superabsorbent Polymer Microspheres Prepared with Hypertonic Saline to Reduce Microsphere Expansion

Cardiovasc Intervent Radiol. 2018 Sep;41(9):1412-1418. doi: 10.1007/s00270-018-1990-4. Epub 2018 May 30.

Abstract

Purpose: To analyze size changes of superabsorbent polymer (SAP) microspheres with the reduced expansion technique, and to evaluate pharmacological advantages of transarterial chemoembolization using cisplatin-loaded SAP microspheres with the reduced expansion technique.

Materials and methods: In an in vitro study, diluted contrast materials containing different concentrations of sodium ions were examined to expand SAP microspheres and determined the reduced expansion technique. Size distributions of cisplatin-loaded SAP microspheres were analyzed. In an in vivo study, TACE was performed using cisplatin-loaded SAP microspheres with the reduced expansion and control techniques in 18 VX2 rabbits.

Results: The degree of expansion was reduced to the greatest extent by using a mixture of non-ionic contrast material and 10% NaCl at a 4:1 ratio. The mean diameter of the reduced expansion of cisplatin-loaded SAP microspheres was 188.4 μm, while that of the control expansion was 404.9 μm. The plasma platinum concentrations of the reduced expansion group at 5 min after TACE were significantly higher than those of the control expansion group (2.19 ± 0.77 vs. 0.75 ± 0.08 μg/mL, P = .01). The tumor platinum concentrations of the reduced expansion group at 1 h were significantly higher than those of the control expansion group (10.76 ± 2.57 vs. 1.57 ± 0.14 μg/g, P = .044).

Conclusion: The expanding level of SAP microspheres can be reduced by using hypertonic saline. Cisplatin-loaded SAP microspheres with the reduced expansion technique have the advantages of achieving higher cisplatin tissue concentration in TACE for liver tumors.

Keywords: Cisplatin; Drug-eluting microsphere; TACE.

MeSH terms

  • Animals
  • Antineoplastic Agents / administration & dosage
  • Antineoplastic Agents / pharmacokinetics
  • Chemoembolization, Therapeutic / methods*
  • Cisplatin / administration & dosage
  • Cisplatin / pharmacokinetics*
  • Contrast Media*
  • Fluoroscopy
  • Liver Neoplasms, Experimental / diagnostic imaging
  • Liver Neoplasms, Experimental / therapy*
  • Male
  • Microspheres*
  • Polymers
  • Rabbits
  • Radiography, Interventional / methods
  • Saline Solution, Hypertonic*

Substances

  • Antineoplastic Agents
  • Contrast Media
  • Polymers
  • Saline Solution, Hypertonic
  • Cisplatin