Visualizing the Brain's Astrocytes with Diverse Chemical Scaffolds

ACS Chem Biol. 2018 Jun 15;13(6):1493-1498. doi: 10.1021/acschembio.8b00391. Epub 2018 May 9.

Abstract

Astrocytes are the most abundant cells in the brain. They support neurons, adjust synaptic strength, and modulate neuronal signaling, yet the full extent of their functions is obscured by the dearth of methods for their visualization and analysis. Here, we report a chemical reporter that targets small molecules specifically to astrocytes both in vitro and in vivo. Fluorescent versions of this tag are imported through an organic cation transporter to label glia across species. The structural modularity of this approach will enable wide-ranging applications for understanding astrocyte biology.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Astrocytes / metabolism*
  • Brain / metabolism*
  • Fluorescence
  • Fluorescent Dyes / chemistry*
  • HEK293 Cells
  • Humans
  • Mice
  • Microscopy, Confocal / methods
  • Pyridinium Compounds / chemistry
  • Rats
  • Rhodamines / chemistry
  • Spinal Cord / metabolism
  • Zebrafish

Substances

  • Fluorescent Dyes
  • Pyridinium Compounds
  • Rhodamines
  • 4-(4-diethylaminostyryl)-N-methylpyridinium