Anthocyanins as a potential pharmacological agent to manage memory deficit, oxidative stress and alterations in ion pump activity induced by experimental sporadic dementia of Alzheimer's type

J Nutr Biochem. 2018 Jun:56:193-204. doi: 10.1016/j.jnutbio.2018.02.014. Epub 2018 Feb 27.

Abstract

Anthocyanins (ANT) are polyphenolic flavonoids with antioxidant and neuroprotective properties. This study evaluated the effect of ANT treatment on cognitive performance and neurochemical parameters in an experimental model of sporadic dementia of Alzheimer's type (SDAT). Adult male rats were divided into four groups: control (1 ml/kg saline, once daily, by gavage), ANT (200 mg/kg, once daily, by gavage), streptozotocin (STZ, 3 mg/kg) and STZ plus ANT. STZ was administered via bilateral intracerebroventricular (ICV) injection (5 μl). ANT were administered after ICV injection for 25 days. Cognitive deficits (short-term memory and spatial memory), oxidative stress parameters, and acetylcholinesterase (AChE) and Na+-K+-ATPase activity in the cerebral cortex and hippocampus were evaluated. ANT treatment protected against the worsening of memory in STZ-induced SDAT. STZ promoted an increase in AChE and Na+-K+-ATPase total and isoform activity in both structures; ANT restored this change. STZ administration induced an increase in lipid peroxidation and decrease in the level of antioxidant enzymes, such as superoxide dismutase (SOD), catalase (CAT) and glutathione peroxidase (GPx), in the cerebral cortex; ANT significantly attenuated these effects. In the hippocampus, an increase in reactive oxygen species (ROS), nitrite and lipid peroxidation levels, and SOD activity and a decrease in CAT and GPx activity were seen after STZ injection. ANT protected against the changes in ROS and antioxidant enzyme levels. In conclusion, the present study showed that treatment with ANT attenuated memory deficits, protected against oxidative damage in the brain, and restored AChE and ion pump activity in an STZ-induced SDAT in rats.

Keywords: Acetylcholinesterase; Alzheimer disease; Anthocyanins; Na(+)-K(+)-ATPase; Oxidative stress; Streptozotocin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcholinesterase / metabolism
  • Alzheimer Disease / chemically induced
  • Alzheimer Disease / drug therapy*
  • Animals
  • Anthocyanins / pharmacology*
  • Antioxidants / therapeutic use
  • Brain / metabolism
  • Catalase / metabolism
  • Cerebral Cortex / metabolism
  • Cognition
  • Disease Models, Animal
  • Glutathione Peroxidase / metabolism
  • Hippocampus / metabolism
  • Infusions, Intraventricular
  • Ion Pumps / metabolism*
  • Lipid Peroxidation
  • Male
  • Maze Learning
  • Memory / drug effects
  • Memory Disorders / chemically induced
  • Memory Disorders / drug therapy*
  • Neuroprotective Agents / therapeutic use
  • Oxidative Stress*
  • Rats
  • Rats, Wistar
  • Streptozocin / adverse effects
  • Sulfhydryl Compounds
  • Superoxide Dismutase / metabolism

Substances

  • Anthocyanins
  • Antioxidants
  • Ion Pumps
  • Neuroprotective Agents
  • Sulfhydryl Compounds
  • Streptozocin
  • Catalase
  • Glutathione Peroxidase
  • Superoxide Dismutase
  • Acetylcholinesterase