Synergistic effects of simvastatin and bone marrow-derived mesenchymal stem cells on hepatic fibrosis

Biochem Biophys Res Commun. 2018 Feb 26;497(1):264-271. doi: 10.1016/j.bbrc.2018.02.067. Epub 2018 Feb 8.

Abstract

The beneficial effects of simvastatin on fibrosis in various organs have been reported. In addition, bone marrow (BM)-derived mesenchymal stem cells (MSCs) have been suggested as an effective therapy for hepatic fibrosis and cirrhosis. Recent evidence suggests that pharmacological treatment devoted to regulating stem cell function is a potential new therapeutic strategy that is drawing nearer to clinical practice. The aim of this study was to determine whether the combination treatment of simvastatin plus MSCs (Sim-MSCs) could have a synergistic effect on hepatic fibrosis in a thioacetamide (TAA)-induced cirrhotic rat model and hepatic stellate cells (HSCs). Cirrhotic livers from rats treated with Sim-MSCs exhibited histological improvement compared to those treated with simvastatin alone. Sim-MSCs combination treatment decreased hepatic collagen distribution, lowered the hydroxyproline content, and rescued liver function impairment in rats with TAA-induced cirrhosis. These protective effects were more potent with Sim-MSCs than with simvastatin alone. The upregulation of collagen-1, α-smooth muscle actin (α-SMA), transforming growth factor (TGF)-β1, and phospho-Smad3 in cirrhotic livers was prevented by the administration of Sim-MSCs. Intriguingly, Sim-MSCs inhibited both TGF-β/Smad3 signaling and α-SMA in HSCs. The Sim-MSCs combination treatment exerted strong protective effects against hepatic fibrosis by suppressing TGF-β/Smad signaling. Simvastatin could act synergistically with MSCs as an efficient therapeutic approach for intractable cirrhosis.

Keywords: Hepatic fibrosis; Liver regeneration; Mesenchymal stem cells; Simvastatin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Bone Marrow Transplantation / methods*
  • Cells, Cultured
  • Combined Modality Therapy / methods
  • Drug Synergism
  • Liver Cirrhosis / pathology
  • Liver Cirrhosis / physiopathology*
  • Liver Cirrhosis / therapy*
  • Liver Function Tests
  • Male
  • Mesenchymal Stem Cell Transplantation / methods*
  • Rats
  • Rats, Sprague-Dawley
  • Simvastatin / administration & dosage*
  • Treatment Outcome

Substances

  • Simvastatin