Synthesis of Bifunctional Thiophenes via Fiesselmann Condensation of Ynone Trifluoroborate Salts

Org Lett. 2018 Jan 5;20(1):198-200. doi: 10.1021/acs.orglett.7b03558. Epub 2017 Dec 14.

Abstract

Ynone trifluoroborate salts undergo a base-promoted condensation reaction with alkylthiols to generate thiophene boronates with complete regiocontrol. The products are isolated in high yield and can be further derivatized through conventional C-B bond functionalization reactions.

Publication types

  • Research Support, Non-U.S. Gov't