Analysis of factors predicting the response to tolvaptan in patients with liver cirrhosis and hepatic edema

J Gastroenterol Hepatol. 2018 Jun;33(6):1256-1263. doi: 10.1111/jgh.14047. Epub 2018 Feb 19.

Abstract

Background and aim: This study aimed to clarify the factors predictive of treatment response to tolvaptan (V2-receptor antagonist) for cirrhotic patients with hepatic edema in a real-world setting.

Methods: In this retrospective, multicenter study, tolvaptan was orally administered at a dose of 7.5 mg once a day. Patients with a decrease in body weight of 1.5 kg or greater from baseline were characterized as responders at day 7.

Results: Of 229 patients, 210 were subjected to this analysis. Patients consisted of 133 men and 77 women, with the median age of 67 years (range, 40-89 years). According to the Child-Pugh classification, five patients were classified as class A, 90 as class B, and 115 as class C. The frequencies of responders and nonresponders were 55.2% and 44.8%, respectively. Blood urea nitrogen (BUN) level was significantly lower in responders compared with nonresponders (P = 3.77 × 10-3 ). Using the receiver operating characteristic curve, the cutoff value of 28.2 mg/dL was the most useful in discriminating responders from nonresponders. Among 154 patients with BUN level of less than 28.2 mg/dL, 95 (61.7%) were responders. By contrast, among 56 patients with BUN level of 28.2 mg/dL or more, 21 (37.5%) were nonresponders (P = 2.70 × 10-3 ). On multivariate analysis, BUN level of <28.2 mg/dL and urine sodium >51 mEq/day were found to be independent factors associated with the response to tolvaptan.

Conclusions: This study suggests that BUN level and urinary sodium excretion are closely associated with the response to tolvaptan in cirrhotic patients with hepatic edema.

Keywords: blood urea nitrogen; diuretics; hepatic edema; tolvaptan.

Publication types

  • Multicenter Study

MeSH terms

  • Administration, Oral
  • Adult
  • Aged
  • Aged, 80 and over
  • Animals
  • Benzazepines / administration & dosage*
  • Biomarkers / blood
  • Biomarkers / urine
  • Blood Urea Nitrogen
  • Edema / complications
  • Edema / diagnosis*
  • Edema / drug therapy*
  • Female
  • Humans
  • Liver Cirrhosis / complications
  • Liver Cirrhosis / diagnosis*
  • Liver Cirrhosis / drug therapy*
  • Liver Diseases / complications
  • Liver Diseases / diagnosis*
  • Liver Diseases / drug therapy*
  • Male
  • Middle Aged
  • Retrospective Studies
  • Sodium / urine
  • Tolvaptan
  • Treatment Outcome

Substances

  • Benzazepines
  • Biomarkers
  • Tolvaptan
  • Sodium