Beta-blockade antagonism of tyramine-induced rise in blood pressure

Eur J Clin Pharmacol. 1988;34(3):263-6. doi: 10.1007/BF00540953.

Abstract

The effect beta-adrenoceptor blockade on the pressor response to tyramine has been investigated in 6 healthy volunteers, each submitted to an i.v. tyramine pressor test before and after 7 days of propranolol 40 mg b.d. or indenolol 60 mg o.d. Tyramine was given as i.v. boluses of 1-6 mg, alternating with saline, in a randomized, single blind fashion. Prior to treatment tyramine caused a temporary, dose-dependent increase in systolic and diastolic blood pressure, whilst the heart rate remained unaffected. Both propranolol and indenolol reduced the pressor response to tyramine, as shown by a significant increase in ED15, i.e. the dose of tyramine required to increase systolic blood pressure by 15%.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Adrenergic beta-Antagonists / pharmacology*
  • Adult
  • Blood Pressure / drug effects*
  • Humans
  • Indenes / pharmacology
  • Male
  • Propanolamines / pharmacology
  • Propranolol / pharmacology
  • Random Allocation
  • Tyramine / antagonists & inhibitors*
  • Vasodilation / drug effects

Substances

  • Adrenergic beta-Antagonists
  • Indenes
  • Propanolamines
  • indenolol
  • Propranolol
  • Tyramine