Nanofiber-based sutures induce endogenous antimicrobial peptide

Nanomedicine (Lond). 2017 Nov;12(21):2597-2609. doi: 10.2217/nnm-2017-0161. Epub 2017 Sep 29.

Abstract

Aim: The aim of this study was to develop nanofiber-based sutures capable of inducing endogenous antimicrobial peptide production.

Methods: We used co-axial electrospinning deposition and rolling to fabricate sutures containing pam3CSK4 peptide and 25-hydroxyvitamin D3 (25D3).

Results: The diameters and mechanical properties of the sutures were adjustable to meet the criteria of United States Pharmacopeia designation. 25D3 exhibited a sustained release from nanofiber sutures over 4 weeks. Pam3CSK4 peptide also showed an initial burst followed by a sustained release over 4 weeks. The co-delivery of 25D3 and pam3CSK4 peptide enhanced cathelicidin antimicrobial peptide production from U937 cells and keratinocytes compared with 25D3 delivery alone. In addition, the 25D3/pam3CSK4 peptide co-loaded nanofiber sutures did not significantly influence proliferation of keratinocytes, fibroblasts, or the monocytic cell lines U937 and HL-60.

Conclusion: The use of 25D3/pam3CSK4 peptide co-loaded nanofiber sutures could potentially induce endogenous antimicrobial peptide production and reduce surgical site infections.

Keywords: 25-hydroxyvitamin D3; co-delivery; electrospun nanofibers; pam3Cys-Ser-(Lys)4 peptide; surgical site infection; sutures.

MeSH terms

  • Antimicrobial Cationic Peptides / biosynthesis*
  • Biomechanical Phenomena
  • Calcifediol / chemistry
  • Calcifediol / pharmacology*
  • Cathelicidins
  • Cell Line
  • Cell Proliferation
  • Drug Carriers
  • Drug Liberation
  • Fibroblasts / cytology
  • Fibroblasts / metabolism
  • Humans
  • Keratinocytes / cytology
  • Keratinocytes / metabolism
  • Lipopeptides / chemistry
  • Lipopeptides / pharmacology*
  • Nanofibers / chemistry*
  • Particle Size
  • Skin / metabolism
  • Surface Properties
  • Sutures*

Substances

  • Antimicrobial Cationic Peptides
  • Drug Carriers
  • Lipopeptides
  • Pam(3)CSK(4) peptide
  • Calcifediol
  • Cathelicidins