Association of the atrial natriuretic factor receptor with guanylate cyclase in solubilized rat glomerular membranes

Biochem Biophys Res Commun. 1987 May 29;145(1):257-62. doi: 10.1016/0006-291x(87)91314-3.

Abstract

The elution profile of solubilized rat glomerular membranes from a gel filtration column showed two peaks of 125I-ANF (atrial natriuretic factor) binding (367 +/- 21, 156 +/- 12 KDa). Over 85% of the total binding for the extract was in the 367 KDa peak. Guanylate cyclase activity was correlated with 125I-ANF specific binding. ANF activation of guanylate cyclase was also observed. As observed previously with particulate membrane, Scatchard-analysis of ANF binding data with the solubilized extract was consistent with a two-site model. Both affinities (Kd's), 4 pM and 1 nM, are within the range of blood concentrations reported for ANF. These observations suggest that most rat glomerular ANF receptors are large molecular complexes coupled with guanylate cyclase in the 300-350 KDa size range.

MeSH terms

  • Animals
  • Atrial Natriuretic Factor / metabolism*
  • Cell Membrane / metabolism
  • Chromatography, Gel
  • Guanylate Cyclase / metabolism*
  • Kidney Glomerulus / metabolism*
  • Kinetics
  • Male
  • Rats
  • Rats, Inbred Strains
  • Receptors, Atrial Natriuretic Factor
  • Receptors, Cell Surface / isolation & purification
  • Receptors, Cell Surface / metabolism*

Substances

  • Receptors, Cell Surface
  • atrial natriuretic peptide, rat
  • Atrial Natriuretic Factor
  • Guanylate Cyclase
  • Receptors, Atrial Natriuretic Factor