Modulation of Salmonella Tumor-Colonization and Intratumoral Anti-angiogenesis by Triptolide and Its Mechanism

Theranostics. 2017 Jun 1;7(8):2250-2260. doi: 10.7150/thno.18816. eCollection 2017.

Abstract

The weakened tumour colonization of attenuated Salmonella has severely hampered its clinical development. In this study, we investigated whether an anti-inflammation and antiangiogenesis compound triptolide could improve the efficacy of VNP20009, a highly attenuated Salmonella strain, against mice melanoma. By comparing the effects of conventional VNP20009 monotherapy and a combination therapy that uses both triptolide and VNP20009, we found that triptolide significantly improved the tumour colonization of VNP20009 by reducing the number of infiltrated neutrophils in the melanoma, which led to a larger necrotic area in the melanoma. Moreover, the combination therapy suppressed tumour angiogenesis by reducing the expression of VEGF in a synergistic manner, retarding the growth of the melanoma. Our study revealed that triptolide could significantly enhance the antitumour effect of VNP20009 by modulating tumour angiogenesis and the host immune response, providing a new understanding of the strategy to improve Salmonella-mediated tumour therapy.

Keywords: Salmonella-mediated tumor therapy; angiogenesis.; melanoma; neutrophils.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biological Therapy / methods
  • Combined Modality Therapy / methods
  • Disease Models, Animal
  • Diterpenes / metabolism*
  • Diterpenes / pharmacology*
  • Epoxy Compounds / metabolism
  • Epoxy Compounds / pharmacology
  • Immunosuppressive Agents / metabolism*
  • Immunosuppressive Agents / pharmacology*
  • Melanoma / microbiology
  • Melanoma / pathology
  • Melanoma / therapy*
  • Mice, Inbred C57BL
  • Necrosis
  • Neovascularization, Pathologic / drug therapy
  • Neutrophils / immunology
  • Phenanthrenes / metabolism*
  • Phenanthrenes / pharmacology*
  • Salmonella / drug effects*
  • Salmonella / growth & development*
  • Treatment Outcome
  • Vascular Endothelial Growth Factor A / antagonists & inhibitors

Substances

  • Diterpenes
  • Epoxy Compounds
  • Immunosuppressive Agents
  • Phenanthrenes
  • Vascular Endothelial Growth Factor A
  • triptolide