Reciprocal modulation of helper Th1 and Th17 cells by the β2-adrenergic receptor agonist drug terbutaline

FEBS J. 2017 Sep;284(18):3018-3028. doi: 10.1111/febs.14166. Epub 2017 Aug 8.

Abstract

Catecholamine hormones are powerful regulators of the immune system produced by the sympathetic nervous system (SNS). They regulate the adaptive immune system by altering T-cell differentiation into T helper (Th) 1 and Th2 cell subsets, but the effect on Th17 cells is not known. Th17 cells, defined, in part, by chemokine receptor CCR6 and cytokine interleukin (IL)-17A, are crucial for mediating certain pathogen-specific responses and are linked with several autoimmune diseases. We demonstrated that a proportion of human Th17 cells express beta 2-adrenergic receptor (β2AR), a G protein-coupled receptor that responds to catecholamines. Activation of peripheral blood mononuclear cells, which were obtained from venous blood drawn from healthy volunteers, with anti-cluster of differentiation 3 (CD3) and anti-CD28 and with a β2-agonist drug, terbutaline (TERB), augmented IL-17A levels (P < 0.01) in the majority of samples. TERB reduced interferon gamma (IFNγ) indicating that IL-17A and IFNγ are reciprocally regulated. Similar reciprocal regulation was observed with dbcAMP. Proliferation of Th cells was monitored by carboxyfluorescein diacetate N-succinimidyl ester labeling and flow cytometry with antibody staining for CD3 and CD4. TERB increased proliferation by a small but significant margin (P < 0.001). Next, Th17 cells (CD4+ CXCR3- CCR6+ ) were purified using an immunomagnetic positive selection kit, which removes all other mononuclear cells. TERB increased IL-17A from purified Th17 cells, which argues that TERB acts directly on Th17 cells. Thus, hormone signals from the SNS maintain a balance of Th cells subtypes through the β2AR.

Keywords: IL-17A; T helper cells; beta 2 adrenergic receptor; norepinephrine; terbutaline.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenergic beta-2 Receptor Agonists / pharmacology*
  • Antibodies, Monoclonal / pharmacology
  • Bucladesine / immunology
  • CD28 Antigens / antagonists & inhibitors
  • CD28 Antigens / genetics
  • CD28 Antigens / immunology
  • CD3 Complex / genetics
  • CD3 Complex / immunology
  • Cell Separation
  • Gene Expression Regulation
  • Humans
  • Interferon-gamma / genetics
  • Interferon-gamma / immunology
  • Interleukin-17 / genetics*
  • Interleukin-17 / immunology
  • Primary Cell Culture
  • Receptors, Adrenergic, beta-2 / genetics*
  • Receptors, Adrenergic, beta-2 / immunology
  • Signal Transduction
  • Terbutaline / pharmacology*
  • Th1 Cells / cytology
  • Th1 Cells / drug effects*
  • Th1 Cells / immunology
  • Th17 Cells / cytology
  • Th17 Cells / drug effects*
  • Th17 Cells / immunology

Substances

  • Adrenergic beta-2 Receptor Agonists
  • Antibodies, Monoclonal
  • CD28 Antigens
  • CD3 Complex
  • IL17A protein, human
  • Interleukin-17
  • Receptors, Adrenergic, beta-2
  • Bucladesine
  • Interferon-gamma
  • Terbutaline