(+)-4-Propyl-9-hydroxynaphthoxazine (PHNO), a new dopaminomimetic, in treatment of parkinsonism

Lancet. 1985 Dec 14;2(8468):1330-1. doi: 10.1016/s0140-6736(85)92627-3.

Abstract

PHNO is a naphthoxazine compound with selective D2 agonist properties and a molecular structure unrelated to the morphine and ergot derivatives that have been used to treat Parkinson's disease. A double-blind, dose-ranging study on 8 patients showed that it is effective in the treatment of parkinsonism; its duration of effect of up to 6 h could make it useful for patients who experience wearing-off reactions with levodopa.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Clinical Trials as Topic
  • Dopamine / physiology
  • Double-Blind Method
  • Female
  • Humans
  • Male
  • Middle Aged
  • Oxazines / adverse effects
  • Oxazines / therapeutic use*
  • Parkinson Disease / drug therapy*
  • Parkinson Disease / physiopathology
  • Time Factors

Substances

  • Oxazines
  • naxagolide
  • Dopamine