Gene-modified NK-92MI cells expressing a chimeric CD16-BB-ζ or CD64-BB-ζ receptor exhibit enhanced cancer-killing ability in combination with therapeutic antibody

Oncotarget. 2017 Jun 6;8(23):37128-37139. doi: 10.18632/oncotarget.16201.

Abstract

Natural killer (NK) cells play a pivotal role in monoclonal antibody-mediated immunotherapy through the antibody-dependent cell-mediated cytotoxicity (ADCC) mechanism. NK-92MI is an interleukin-2 (IL-2)-independent cell line, which was derived from NK-92 cells with superior cytotoxicity toward a wide range of tumor cells in vitro and in vivo. Nonetheless, the Fc-receptor (CD16) that usually mediates ADCC is absent in NK-92 and NK-92MI cells. To apply NK-92MI cell-based immunotherapy to cancer treatment, we designed and generated two chimeric receptors in NK-92MI cells that can bind the Fc portion of human immunoglobulins. The construct includes the low-affinity Fc receptor CD16 (158F) or the high-affinity Fc receptor CD64, with the addition of the CD8a extracellular domain, CD28 transmembrane domains, two costimulatory domains (CD28 and 4-1BB), and the signaling domain from CD3ζ. The resulting chimeric receptors, termed CD16-BB-ζ and CD64-BB-ζ, were used to generate modified NK-92MI cells expressing the chimeric receptor, which were named NK-92MIhCD16 and NK-92MIhCD64 cells, respectively. We found that NK-92MIhCD16 and NK-92MIhCD64 cells significantly improved cytotoxicity against CD20-positive non-Hodgkin's lymphoma cells in the presence of rituximab. These results suggest that the chimeric receptor-expressing NK-92MI cells may enhance the clinical responses to currently available anticancer monoclonal antibodies.

Keywords: NK-92MI; chimeric CD16/CD64-BB-ζ receptor; therapeutic antibody.

MeSH terms

  • Animals
  • Antibody-Dependent Cell Cytotoxicity / drug effects
  • Antibody-Dependent Cell Cytotoxicity / immunology*
  • Antigens, CD20 / immunology
  • Antigens, CD20 / metabolism
  • Antineoplastic Agents, Immunological / immunology
  • Antineoplastic Agents, Immunological / pharmacology
  • Cell Line, Tumor
  • Cell Survival / drug effects
  • Cell Survival / immunology
  • Humans
  • K562 Cells
  • Kaplan-Meier Estimate
  • Killer Cells, Natural / immunology*
  • Killer Cells, Natural / metabolism
  • Lymphoma, Mantle-Cell / drug therapy
  • Lymphoma, Mantle-Cell / immunology
  • Lymphoma, Mantle-Cell / pathology
  • Mice, Inbred NOD
  • Mice, Knockout
  • Receptors, IgG / genetics
  • Receptors, IgG / immunology*
  • Receptors, IgG / metabolism
  • Recombinant Fusion Proteins / genetics
  • Recombinant Fusion Proteins / immunology*
  • Recombinant Fusion Proteins / metabolism
  • Rituximab / immunology
  • Rituximab / pharmacology
  • Xenograft Model Antitumor Assays

Substances

  • Antigens, CD20
  • Antineoplastic Agents, Immunological
  • Receptors, IgG
  • Recombinant Fusion Proteins
  • Rituximab