[The effects of eicosapentaenoic acid ethyl ester (EPA-E) on arterial thrombosis in rabbits and vascular lesions in rats]

Nihon Yakurigaku Zasshi. 1988 Feb;91(2):81-9. doi: 10.1254/fpj.91.81.
[Article in Japanese]

Abstract

The effects of highly purified ethyl ester of eicosapentaenoic acid (EPA-E) on ellagic acid-induced thrombus formation in the stenosed femoral artery in rabbits and on the progression of laurate-induced vascular lesions in rats were examined. (1) EPA-E in single administration significantly prevented the thrombus formation induced by ellagic acid in the stenosed femoral artery of rabbits. (2) EPA-E restored the hypercoagulation activity at 5 min and 3 hr after the ellagic acid injection. Platelet aggregability induced by arachidonic acid decreased at 5 min and 3 hr after the ellagic acid injection; EPA-E had little effect on this change. EPA-E showed almost no effect on fibrinolytic activity, blood viscosity and filterability of washed red blood cells after the ellagic acid injection. (3) Moreover, EPA-E in daily administrations showed a significant preventative effect against the laurate-induced vascular lesions in rats. The efficacy of EPA-E on arterial thrombosis and vascular lesions observed in this study suggests that EPA-E is a candidate for the treatment of peripheral circulatory disturbance.

MeSH terms

  • Animals
  • Eicosapentaenoic Acid / analogs & derivatives*
  • Eicosapentaenoic Acid / pharmacology
  • Ellagic Acid
  • Gangrene / chemically induced
  • Gangrene / prevention & control*
  • Laurates
  • Male
  • Rabbits
  • Rats
  • Rats, Inbred Strains
  • Thrombosis / chemically induced
  • Thrombosis / prevention & control*

Substances

  • Laurates
  • Ellagic Acid
  • eicosapentaenoic acid ethyl ester
  • Eicosapentaenoic Acid