Pentraxin-2 suppresses c-Jun/AP-1 signaling to inhibit progressive fibrotic disease

JCI Insight. 2016 Dec 8;1(20):e87446. doi: 10.1172/jci.insight.87446.

Abstract

Pentraxin-2 (PTX-2), also known as serum amyloid P component (SAP/APCS), is a constitutive, antiinflammatory, innate immune plasma protein whose circulating level is decreased in chronic human fibrotic diseases. Here we show that recombinant human PTX-2 (rhPTX-2) retards progression of chronic kidney disease in Col4a3 mutant mice with Alport syndrome, reducing blood markers of kidney failure, enhancing lifespan by 20%, and improving histological signs of disease. Exogenously delivered rhPTX-2 was detected in macrophages but also in tubular epithelial cells, where it counteracted macrophage activation and was cytoprotective for the epithelium. Computational analysis of genes regulated by rhPTX-2 identified the transcriptional regulator c-Jun along with its activator protein-1 (AP-1) binding partners as a central target for the function of rhPTX-2. Accordingly, PTX-2 attenuates c-Jun and AP-1 activity, and reduces expression of AP-1-dependent inflammatory genes in both monocytes and epithelium. Our studies therefore identify rhPTX-2 as a potential therapy for chronic fibrotic disease of the kidney and an important inhibitor of pathological c-Jun signaling in this setting.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • C-Reactive Protein / pharmacology*
  • Cells, Cultured
  • Fibrosis
  • Humans
  • Kidney / pathology*
  • Macrophage Activation
  • Mice
  • Mice, 129 Strain
  • Mice, Knockout
  • Monocytes
  • Nephritis, Hereditary / pathology
  • Nephritis, Hereditary / therapy*
  • Nerve Tissue Proteins / pharmacology*
  • Proto-Oncogene Proteins c-jun / antagonists & inhibitors*
  • Recombinant Proteins / pharmacology
  • Signal Transduction*
  • Transcription Factor AP-1 / antagonists & inhibitors*

Substances

  • Nerve Tissue Proteins
  • Proto-Oncogene Proteins c-jun
  • Recombinant Proteins
  • Transcription Factor AP-1
  • neuronal pentraxin
  • C-Reactive Protein