The 18 kDa cytosolic acid phosphatase from bovine live has phosphotyrosine phosphatase activity on the autophosphorylated epidermal growth factor receptor

FEBS Lett. 1989 Jul 3;250(2):469-73. doi: 10.1016/0014-5793(89)80778-1.

Abstract

In this paper we demonstrate that the cytosolic low-Mr acid phosphatase purified from bovine liver has phosphotyrosine protein phosphatase activity on 32P-autophosphorylated epidermal growth factor (EGF) receptor. This activity was significantly inhibited by orthovanadate and p-hydroxymercuribenzoate; the latter result indicates that free sulfhydryl groups are required for phosphotyrosine phosphatase activity. The enzyme was active in a broad pH range, with maximum activity between pH 5.5 and 7.5. The apparent Km for 32P-EGF receptor dephosphorylation was 4 nM. The enzyme appeared to be specific for phosphotyrosine in that it dephosphorylated the autophosphorylated EGF receptor and L-phosphotyrosine, but not 32P-Ser-casein, L-phosphoserine or L-phosphothreonine. These data suggest that the cytosolic low-Mr acid phosphatase might play a regulatory role in EGF receptor-dependent transmembrane signalling.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acid Phosphatase / metabolism*
  • Animals
  • Cattle
  • Cytosol / enzymology
  • Electrophoresis, Polyacrylamide Gel
  • Epidermal Growth Factor / metabolism*
  • ErbB Receptors / metabolism*
  • Hydrogen-Ion Concentration
  • Liver / enzymology*
  • Phosphorylation
  • Substrate Specificity

Substances

  • Epidermal Growth Factor
  • ErbB Receptors
  • Acid Phosphatase