Stability of suxamethonium in pharmaceutical solution for injection by validated stability-indicating chromatographic method

J Clin Anesth. 2016 Dec:35:551-559. doi: 10.1016/j.jclinane.2016.09.025. Epub 2016 Oct 23.

Abstract

Study objective: To assess the stability of pharmaceutical suxamethonium (succinylcholine) solution for injection by validated stability-indicating chromatographic method in vials stored at room temperature.

Methods: The chromatographic assay was achieved by using a detector wavelength set at 218 nm, a C18 column, and an isocratic mobile phase (100% of water) at a flow rate of 0.6 mL/min for 5 minutes. The method was validated according to the International Conference on Harmonization guidelines with respect to the stability-indicating capacity of the method including linearity, limits of detection and quantitation, precision, accuracy, system suitability, robustness, and forced degradations.

Results: Linearity was achieved in the concentration range of 5 to 40 mg/mL with a correlation coefficient higher than 0.999. The limits of detection and quantification were 0.8 and 0.9 mg/mL, respectively. The percentage relative standard deviation for intraday (1.3-1.7) and interday (0.1-2.0) precision was found to be less than 2.1%. Accuracy was assessed by the recovery test of suxamethonium from solution for injection (99.5%-101.2%).

Conclusion: Storage of suxamethonium solution for injection vials at ambient temperature (22°C-26°C) for 17 days demonstrated that at least 95% of original suxamethonium concentration remained stable.

Keywords: Forced degradation; Liquid chromatography; Solution for injection; Stability; Stability-indicating; Suxamethonium.

MeSH terms

  • Chromatography, High Pressure Liquid*
  • Drug Stability
  • Neuromuscular Depolarizing Agents / analysis*
  • Neuromuscular Depolarizing Agents / chemistry
  • Pharmaceutical Solutions
  • Reproducibility of Results
  • Succinylcholine / analysis*
  • Succinylcholine / chemistry

Substances

  • Neuromuscular Depolarizing Agents
  • Pharmaceutical Solutions
  • Succinylcholine