Lysosome-mitochondria-mediated apoptosis specifically evoked in cancer cells induced by gold nanorods

Nanomedicine (Lond). 2016 Aug;11(15):1993-2006. doi: 10.2217/nnm-2016-0139. Epub 2016 Jun 3.

Abstract

Aim: The main aim of this article is to explain the apoptosis mechanisms of cancer cells specifically triggered by gold nanorods (GNRs).

Materials & methods: GNRs were synthesized and optimized, the lysosome damage, cathepsin D, mitochondrial membrane potential, caspase-9, cleaved caspase-9, caspase-3 and intracellular GNRs location related to apoptosis was systematically evaluated.

Results: GNRs specifically induce cancer cell apoptosis while posing a negligible impact on normal cells. After incubation with GNRs, the lysosomal permeability in cancer cells as indicated by cathepsin D was markedly higher than that in normal cells and resulted in an obvious decrease in mitochondrial membrane potential. Western blot analysis further confirmed that apoptosis occurred through caspase-9 and caspase-3 activation following mitochondrial damage. Transmission electron microscope images showed that GNRs did not appear in most of the damaged mitochondria but mainly accumulated in lysosomes.

Conclusion: These findings indicated that GNR-induced apoptosis specifically in cancer cells by affecting lysosomes and mitochondria.

Keywords: apoptosis; gold nanorods; lysosome; mitochondrion.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects*
  • Caspase 3 / metabolism
  • Caspase 9 / metabolism
  • Cell Line, Tumor
  • Cell Survival
  • Cricetulus
  • Gold / chemistry*
  • Gold / therapeutic use*
  • Humans
  • Lysosomes / metabolism*
  • Membrane Potential, Mitochondrial
  • Mice
  • Mitochondria / metabolism*
  • Nanotubes / chemistry*
  • Particle Size

Substances

  • Gold
  • Caspase 3
  • Caspase 9