Leptin promotes proliferation and metastasis of human gallbladder cancer through OB-Rb leptin receptor

Int J Oncol. 2016 Jul;49(1):197-206. doi: 10.3892/ijo.2016.3530. Epub 2016 May 18.

Abstract

Emerging evidence has shown that leptin, an adipocyte-derived cytokine that is closely associated with obesity, play a significant role in carcinogenesis and tumorigenesis. However, its impact on gallbladder cancer (GBC) remains unclear. In this study, we firstly found that leptin and its functional receptor OB-Rb were significantly co-expressed in human GBC tissues and cell lines, the content of which were higher than those in normal human gallbladder tissues. Treatment with leptin promoted the proliferation, migration and invasion of GBC cells, which were attenuated by OB-Rb shRNA. Blocking in the G2/M period of cell cycle, increasing of MMP3 and MMP9, increasing of VEGF-C/D, activation of SOCS3/JAK2/p-STAT3 pathway was demonstrated after treatment with leptin. All of these positive responses were attenuated by OB-Rb receptor shRNA. Taken together, our findings suggest that leptin promoted the proliferation, migration and invasion of GBC cells by increasing OB-Rb expression through the SOCS3/JAK2/p-STAT3 signal pathway. Targeting the leptin/OB-Rb axis could be an attractive therapeutic strategy for treatment of GBC.

MeSH terms

  • Cell Movement / genetics
  • Cell Proliferation / genetics*
  • Gallbladder Neoplasms / drug therapy
  • Gallbladder Neoplasms / genetics*
  • Gallbladder Neoplasms / pathology
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Janus Kinase 2 / genetics
  • Leptin / administration & dosage
  • Leptin / genetics*
  • Neoplasm Invasiveness / genetics
  • Neoplasm Metastasis
  • RNA, Small Interfering
  • Receptors, Leptin / biosynthesis
  • Receptors, Leptin / genetics*
  • STAT3 Transcription Factor / genetics
  • Signal Transduction / genetics
  • Suppressor of Cytokine Signaling 3 Protein / genetics
  • Vascular Endothelial Growth Factor C / genetics
  • Vascular Endothelial Growth Factor D / genetics

Substances

  • LEPR protein, human
  • Leptin
  • RNA, Small Interfering
  • Receptors, Leptin
  • SOCS3 protein, human
  • STAT3 Transcription Factor
  • STAT3 protein, human
  • Suppressor of Cytokine Signaling 3 Protein
  • Vascular Endothelial Growth Factor C
  • Vascular Endothelial Growth Factor D
  • JAK2 protein, human
  • Janus Kinase 2