Pharmacokinetics of butorphanol delivered with an osmotic pump during a seven-day period in common peafowl (Pavo cristatus)

Am J Vet Res. 2015 Dec;76(12):1070-6. doi: 10.2460/ajvr.76.12.1070.

Abstract

Objective: To determine pharmacokinetics of butorphanol delivered via osmotic pumps in common peafowl (Pavo cristatus) as a method for analgesic administration to avian species.

Animals: 14 healthy adult male common peafowl.

Procedures: A preliminary experiment was conducted with 2 birds to establish time point and concentration requirements. Then, the remaining 12 birds were anesthetized, and 2 osmotic pumps containing butorphanol (volume, 2 mL; mean dosage, 247 μg/kg/h) were implanted subcutaneously in each bird for 7 days prior to removal. Blood samples were collected before pump implantation (time 0); 3, 6, 12, 24, 48, 72, 96, 120, 144, and 168 hours after pump implantation; and 3 and 6 hours after pump removal. Plasma butorphanol concentrations were measured via liquid chromatography-mass spectrometry.

Results: Plasma concentrations peaked (mean, 106.4 μg/L; range, 61.8 to 133.0 μg/L) at a mean of 39.0 hours, with no evidence of sedation in any bird. After pump removal, butorphanol was rapidly eliminated (half-life, 1.45 hours; range, 1.31 to 1.64 hours; n = 5). Mean clearance per fraction of dose absorbed was 2.89 L/kg/h (range, 2.00 to 5.55 L/kg/h). Mean amount of time the plasma butorphanol concentration was ≥ 60 μg/L was 85.6 hours (range, 3.5 to 155.3 hours).

Conclusions and clinical relevance: Plasma concentrations of butorphanol in common peafowl were maintained at or above reported efficacious analgesic concentrations. This study established a method for administering analgesics to avian patients without the need for frequent handling or injections. Use of these osmotic pumps may provide options for avian analgesia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analgesia
  • Analgesics / administration & dosage
  • Analgesics / blood
  • Analgesics, Opioid / administration & dosage*
  • Analgesics, Opioid / blood
  • Animals
  • Body Weight
  • Butorphanol / administration & dosage*
  • Butorphanol / blood
  • Chromatography, Liquid
  • Galliformes*
  • Half-Life
  • Male
  • Mass Spectrometry
  • Osmosis
  • Pain
  • Time Factors

Substances

  • Analgesics
  • Analgesics, Opioid
  • Butorphanol