Inotropic effects of endothelin in ferret ventricular myocardium

Eur J Pharmacol. 1989 Apr 25;163(2-3):365-7. doi: 10.1016/0014-2999(89)90208-2.

Abstract

The characteristics of the inotropic response to endothelin were studied in isolated ferret papillary muscle preparations. Endothelin (0.1-10 nM) induced concentration-dependent positive inotropic effects. At 10 nM, isometric tension increased by 17%, maximum rate of tension development by 18%, maximum velocity of unloaded shortening by 23% and peak isotonic shortening by 11%. Time to peak isometric tension and half isometric relaxation time were unaltered by endothelin. This pattern of change is similar to that of elevating extracellular calcium concentration.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Carnivora / physiology*
  • Endothelins
  • Ferrets / physiology*
  • Heart / drug effects*
  • In Vitro Techniques
  • Isometric Contraction / drug effects
  • Myocardial Contraction / drug effects*
  • Peptides / pharmacology*

Substances

  • Endothelins
  • Peptides