General Homologation Strategy for Synthesis of L-glycero- and D-glycero-Heptopyranoses

Org Lett. 2015 Nov 20;17(22):5536-9. doi: 10.1021/acs.orglett.5b02620. Epub 2015 Nov 11.

Abstract

A general and stereospecific homologation strategy for the synthesis of heptopyranosides is reported. The strategy employs the Wittig olefination and proline-catalyzed α-aminoxylation to achieve one carbon elongation and stereoselective hydroxylation at the C6 position, respectively. The L-glycero- and D-glycero-heptopyranosides can be obtained with nearly perfect stereoselectivity. Further study reveals the difference in the chemical shift of the C6 proton of L/D-glycero-heptopyranosyl diastereomers, which is found to be useful for assignment of the configuration of heptopyranosides.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Glycosides / chemical synthesis
  • Glycosides / chemistry
  • Heptoses / chemical synthesis*
  • Heptoses / chemistry
  • Molecular Structure
  • Stereoisomerism
  • Structure-Activity Relationship

Substances

  • Glycosides
  • Heptoses