Acute ingestion of citrulline stimulates nitric oxide synthesis but does not increase blood flow in healthy young and older adults with heart failure

Am J Physiol Endocrinol Metab. 2015 Dec 1;309(11):E915-24. doi: 10.1152/ajpendo.00339.2015. Epub 2015 Oct 6.

Abstract

To determine if age-associated vascular dysfunction in older adults with heart failure (HF) is due to insufficient synthesis of nitric oxide (NO), we performed two separate studies: 1) a kinetic study with a stable isotope tracer method to determine in vivo kinetics of NO metabolism, and 2) a vascular function study using a plethysmography method to determine reactive hyperemic forearm blood flow (RH-FBF) in older and young adults in the fasted state and in response to citrulline ingestion. In the fasted state, NO synthesis (per kg body wt) was ∼ 50% lower in older vs. young adults and was related to a decreased rate of appearance of the NO precursor arginine. Citrulline ingestion (3 g) stimulated de novo arginine synthesis in both older [6.88 ± 0.83 to 35.40 ± 4.90 μmol · kg body wt(-1) · h(-1)] and to a greater extent in young adults (12.02 ± 1.01 to 66.26 ± 4.79 μmol · kg body wt(-1) · h(-1)). NO synthesis rate increased correspondingly in older (0.17 ± 0.01 to 2.12 ± 0.36 μmol · kg body wt(-1) · h(-1)) and to a greater extent in young adults (0.36 ± 0.04 to 3.57 ± 0.47 μmol · kg body wt(-1) · h(-1)). Consistent with the kinetic data, RH-FBF in the fasted state was ∼ 40% reduced in older vs. young adults. However, citrulline ingestion (10 g) failed to increase RH-FBF in either older or young adults. In conclusion, citrulline ingestion improved impaired NO synthesis in older HF adults but not RH-FBF, suggesting that factors other than NO synthesis play a role in the impaired RH-FBF in older HF adults, and/or it may require a longer duration of supplementation to be effective in improving RH-FBF.

Keywords: aging; arginine; endothelial dysfunction; stable isotope tracers.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adult
  • Aged
  • Arginine / blood
  • Arginine / metabolism
  • Cardiovascular Agents / adverse effects
  • Cardiovascular Agents / therapeutic use*
  • Citrulline / adverse effects
  • Citrulline / therapeutic use*
  • Dietary Supplements* / adverse effects
  • Elder Nutritional Physiological Phenomena*
  • Endothelium, Vascular / metabolism
  • Endothelium, Vascular / physiopathology
  • Female
  • Forearm
  • Heart Failure / blood
  • Heart Failure / diet therapy*
  • Heart Failure / metabolism
  • Heart Failure / physiopathology
  • Humans
  • Hyperemia / etiology
  • Kinetics
  • Male
  • Middle Aged
  • Nitric Oxide / agonists*
  • Nitric Oxide / blood
  • Nitric Oxide / metabolism
  • Regional Blood Flow
  • Severity of Illness Index
  • Up-Regulation*
  • Young Adult

Substances

  • Cardiovascular Agents
  • Citrulline
  • Nitric Oxide
  • Arginine