The interactions between a small molecule and G-quadruplexes are visualized by fluorescence lifetime imaging microscopy

Nat Commun. 2015 Sep 9:6:8178. doi: 10.1038/ncomms9178.

Abstract

Guanine-rich oligonucleotides can fold into quadruple-stranded helical structures known as G-quadruplexes. Mounting experimental evidence has gathered suggesting that these non-canonical nucleic acid structures form in vivo and play essential biological roles. However, to date, there are no small-molecule optical probes to image G-quadruplexes in live cells. Herein, we report the design and development of a small fluorescent molecule, which can be used as an optical probe for G-quadruplexes. We demonstrate that the fluorescence lifetime of this new probe changes considerably upon interaction with different nucleic acid topologies. Specifically, longer fluorescence lifetimes are observed in vitro for G-quadruplexes than for double- and single-stranded nucleic acids. Cellular studies confirm that this molecule is cell permeable, has low cytotoxicity and localizes primarily in the cell nucleus. Furthermore, using fluorescence lifetime imaging microscopy, live-cell imaging suggests that the probe can be used to study the interaction of small molecules with G-quadruplexes in vivo.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line, Tumor
  • Fluorescent Dyes*
  • G-Quadruplexes*
  • Humans
  • In Vitro Techniques
  • Intravital Microscopy
  • Microscopy, Confocal
  • Microscopy, Fluorescence
  • Nucleic Acid Conformation
  • Oligonucleotides*
  • Spectrometry, Fluorescence

Substances

  • Fluorescent Dyes
  • Oligonucleotides