Targeting MYC Translation in Colorectal Cancer

Cancer Discov. 2015 Jul;5(7):701-3. doi: 10.1158/2159-8290.CD-15-0660.

Abstract

There is a great interest in finding ways to inhibit the expression or activity of the "undruggable" MYC, a master regulator of transcription and one of the most deadly oncoproteins in human cancer. In this issue of Cancer Discovery, Wiegering and colleagues find a way of inhibiting translation of MYC in colorectal cancer cells by directly targeting the translation initiation factor eIF4A, resulting in inhibition of MYC-dependent proliferation of colorectal tumor cells in vitro and in vivo.

Publication types

  • Comment

MeSH terms

  • Animals
  • Antineoplastic Agents / administration & dosage*
  • Colorectal Neoplasms / drug therapy*
  • Colorectal Neoplasms / genetics*
  • Humans
  • Peptide Chain Initiation, Translational / drug effects*
  • Proto-Oncogene Proteins c-myc / genetics*
  • Triterpenes / administration & dosage*

Substances

  • Antineoplastic Agents
  • Proto-Oncogene Proteins c-myc
  • Triterpenes