Polydatin: a new therapeutic agent against multiorgan dysfunction

J Surg Res. 2015 Sep;198(1):192-9. doi: 10.1016/j.jss.2015.05.041. Epub 2015 May 27.

Abstract

Background: Polydatin (PD), a monocrystalline and polyphenolic drug isolated from a traditional Chinese herb (Polygonum cuspidatum), is protective against mitochondrial dysfunction and has been approved for clinical trials in the treatment of shock. However, whether the administration of PD has a therapeutic effect on multiple-organ dysfunction syndrome (MODS) requires investigation.

Material and methods: MODS was induced in Sprague-Dawley rats via hemorrhage and ligation and puncture of cecum-induced sepsis. The rats were divided into three groups as follows: MODS + PD, MODS + normal saline, and a control group (no treatment). Survival time, blood biochemical indexes, and histopathologic changes in various organs were evaluated; serum oxidative stress (advanced oxidative protein products [AOPPs]) and proinflammatory cytokines (tumor necrosis factor-α, interleukin 1β, and interleukin 6) were assayed using enzyme-linked immunosorbent assay. Apoptosis-related protein expression (B-cell lymphoma-2 [Bcl-2] and Bax) was assayed by immunohistochemical and Western blotting methods, whereas caspase-3 activity was assayed by spectrophotometry.

Results: PD improved organ function, prolonged survival time, and reduced MODS incidence and serum levels of AOPPs and proinflammatory cytokines. It also decreased Bax levels and caspase-3 activity and increased Bcl-2 levels in the kidney and liver.

Conclusions: PD may serve as a potential therapeutic for MODS, as it suppresses oxidative stress, inhibits inflammatory response, attenuates apoptosis, and protects against mitochondrial dysfunction.

Keywords: Apoptosis; Inflammation; Multiorgan dysfunction syndrome; Oxidative stress; Polydatin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Caspase 3 / metabolism
  • Cytokines / blood
  • Female
  • Glucosides / therapeutic use*
  • Multiple Organ Failure / drug therapy*
  • Multiple Organ Failure / immunology
  • Multiple Organ Failure / mortality
  • Proto-Oncogene Proteins c-bcl-2 / analysis
  • Rats
  • Rats, Sprague-Dawley
  • Stilbenes / therapeutic use*

Substances

  • Cytokines
  • Glucosides
  • Proto-Oncogene Proteins c-bcl-2
  • Stilbenes
  • Casp3 protein, rat
  • Caspase 3
  • polydatin