Optimal single-dose epidural neostigmine for postoperative analgesia after partial hepatectomy

Indian J Pharmacol. 2014 Nov-Dec;46(6):613-6. doi: 10.4103/0253-7613.144918.

Abstract

Objective: Neostigmine can produce analgesia by acting on the spinal cord. This study was to determine the optimal single-dose of epidural neostigmine for postoperative analgesia after partial hepatectomy.

Patients and methods: Twenty-six patients undergoing elective partial hepatectomy under general anesthesia combined with epidural block were studied. The dose of epidural neostigmine was determined using Dixon's up-and-down method, starting from neostigmine 100 μg with an interval of 25 μg. Thirty minutes after skin incision, a predetermined dose of neostigmine was injected via the epidural catheter. Each patient received 0.125% bupivacaine and fentanyl 2 μg/ml for patient controlled epidural analgesia (PCEA) after the operation. Assessment of analgesia quality was performed at 8 h and 24 h after the operation.

Results: The ED50 of epidural neostigmine in combination with PCEA for satisfactory analgesia was 226.78 ± 33.20 μg. Probit analysis showed that the ED50 and ED95 of epidural neostigmine were 228.63 μg (95% CI = 197.95-299.77 μg) and 300.12 μg (95% CI = 259.44-741.65 μg), respectively.

Conclusion: The ED50 and ED95 of epidural neostigmine in combination with PCEA for satisfactory analgesia after partial hepatectomy were 228.63 μg (95% CI = 197.95-299.77 μg) and 300.12 μg (95% CI = 259.44-741.65 μg).

Keywords: Dixon's up-and-down method; neostigmine; optimal dose; patient controlled epidural analgesia; postoperative analgesia.

Publication types

  • Clinical Trial

MeSH terms

  • Adolescent
  • Adult
  • Analgesia, Epidural*
  • Analgesia, Patient-Controlled*
  • Analgesics / administration & dosage*
  • Analgesics / therapeutic use
  • Dose-Response Relationship, Drug
  • Female
  • Hepatectomy*
  • Humans
  • Injections, Epidural
  • Male
  • Middle Aged
  • Neostigmine / administration & dosage*
  • Neostigmine / therapeutic use
  • Young Adult

Substances

  • Analgesics
  • Neostigmine