Hepatic miR-378 targets p110α and controls glucose and lipid homeostasis by modulating hepatic insulin signalling

Nat Commun. 2014 Dec 4:5:5684. doi: 10.1038/ncomms6684.

Abstract

Understanding the regulation of insulin signalling in tissues provides insights into carbohydrate and lipid metabolism in physiology and disease. Here we show that hepatic miR-378/378* expression changes in response to fasting and refeeding in mice. Mice overexpressing hepatic miR-378/378* exhibit pure hepatic insulin resistance. miR-378 inhibits hepatic insulin signalling through targeting p110α, a subunit of PI3K and hence a critical component of insulin signalling. Knockdown of hepatic p110α mimics the effect of miR-378, while restoration of p110α expression abolishes the action of miR-378 on insulin signalling as well as its systemic effects on glucose and lipid homeostasis. miR-378/378* knockout mice display hypoglycemia and increased hepatic triglyceride level with enhanced insulin sensitivity. Inhibition of hepatic p110α in miR-378/378* knockout mice corrects the abnormal glucose tolerance. Finally, we show that overexpression of hepatic miR-378/378* ameliorates hepatic steatosis in ob/ob mice without exacerbating hyperglycemia. Our findings establish fasting-responsive miR-378 as a critical regulator of hepatic insulin signalling.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blood Glucose / metabolism*
  • Class I Phosphatidylinositol 3-Kinases
  • Fasting / metabolism
  • Fatty Liver / genetics
  • Fatty Liver / metabolism
  • Glucose / metabolism
  • Glucose Intolerance / genetics*
  • Glucose Intolerance / metabolism
  • Homeostasis
  • Insulin / metabolism*
  • Insulin Resistance / genetics*
  • Lipid Metabolism / genetics*
  • Liver / metabolism*
  • Mice
  • Mice, Knockout
  • Mice, Obese
  • MicroRNAs / genetics*
  • Phosphatidylinositol 3-Kinases / genetics*
  • Phosphatidylinositol 3-Kinases / metabolism
  • Signal Transduction

Substances

  • Blood Glucose
  • Insulin
  • MIRN378 microRNA, mouse
  • MicroRNAs
  • Class I Phosphatidylinositol 3-Kinases
  • Pik3ca protein, mouse
  • Glucose