IL-1 induces rapid phosphorylation of the IL-1 receptor

J Immunol. 1989 Nov 15;143(10):3235-40.

Abstract

The IL-1R on murine T cells is a Mr = 80,000 plasma membrane glycoprotein. cDNA cloning and transfection experiments have shown that this is an integral membrane protein, which binds both IL-1 alpha and IL-1 beta and transduces the IL-1 signal. A mAb, RM-5, which binds an epitope on the receptor which is distinct from the IL-1 binding site has been produced in rats. RM-5 has been used to immunoprecipitate the IL-1R from 32P-orthophosphate labeled CHO cells which express approximately 100,000 functional, murine rIL-1R/cell. Phosphorylation of the receptor was observed as early as 1 min after the addition of IL-1 and continued for periods of up to 30 min. Phosphorylation increases as the concentration of IL-1 increases from 10(-13) to 10(-8) M. Potassium hydroxide hydrolysis of the phosphorylated IL-1R shows that more than 90% of the phosphate is incorporated into serine or threonine. Thus, one of the earliest events after IL-1 binding to the IL-1R is activation of a serine/threonine protein kinase and phosphorylation of the IL-1R itself.

MeSH terms

  • Animals
  • Antibodies, Monoclonal / analysis
  • Antibody Specificity
  • Binding Sites, Antibody
  • Cell Line
  • Dose-Response Relationship, Immunologic
  • Humans
  • Interleukin-1 / metabolism
  • Interleukin-1 / pharmacology*
  • Kinetics
  • Phosphoproteins / isolation & purification
  • Phosphorylation
  • Rats
  • Receptors, Immunologic / biosynthesis
  • Receptors, Immunologic / metabolism*
  • Receptors, Interleukin-1

Substances

  • Antibodies, Monoclonal
  • Interleukin-1
  • Phosphoproteins
  • Receptors, Immunologic
  • Receptors, Interleukin-1