Liver Med23 ablation improves glucose and lipid metabolism through modulating FOXO1 activity

Cell Res. 2014 Oct;24(10):1250-65. doi: 10.1038/cr.2014.120. Epub 2014 Sep 16.

Abstract

Mediator complex is a molecular hub integrating signaling, transcription factors, and RNA polymerase II (RNAPII) machinery. Mediator MED23 is involved in adipogenesis and smooth muscle cell differentiation, suggesting its role in energy homeostasis. Here, through the generation and analysis of a liver-specific Med23-knockout mouse, we found that liver Med23 deletion improved glucose and lipid metabolism, as well as insulin responsiveness, and prevented diet-induced obesity. Remarkably, acute hepatic Med23 knockdown in db/db mice significantly improved the lipid profile and glucose tolerance. Mechanistically, MED23 participates in gluconeogenesis and cholesterol synthesis through modulating the transcriptional activity of FOXO1, a key metabolic transcription factor. Indeed, hepatic Med23 deletion impaired the Mediator and RNAPII recruitment and attenuated the expression of FOXO1 target genes. Moreover, this functional interaction between FOXO1 and MED23 is evolutionarily conserved, as the in vivo activities of dFOXO in larval fat body and in adult wing can be partially blocked by Med23 knockdown in Drosophila. Collectively, our data revealed Mediator MED23 as a novel regulator for energy homeostasis, suggesting potential therapeutic strategies against metabolic diseases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cells, Cultured
  • Cholesterol / biosynthesis
  • Drosophila / growth & development
  • Drosophila Proteins / antagonists & inhibitors
  • Drosophila Proteins / genetics
  • Drosophila Proteins / metabolism
  • Forkhead Box Protein O1
  • Forkhead Transcription Factors / deficiency
  • Forkhead Transcription Factors / genetics
  • Forkhead Transcription Factors / metabolism*
  • Gluconeogenesis
  • Glucose / metabolism*
  • Hepatocytes / cytology
  • Hepatocytes / metabolism
  • Insulin / metabolism
  • Larva / metabolism
  • Lipid Metabolism / genetics*
  • Liver / metabolism*
  • Male
  • Mediator Complex / antagonists & inhibitors
  • Mediator Complex / genetics*
  • Mediator Complex / metabolism
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Mice, Obese
  • RNA Interference
  • RNA Polymerase II / metabolism
  • Signal Transduction
  • Transcription, Genetic

Substances

  • Drosophila Proteins
  • Forkhead Box Protein O1
  • Forkhead Transcription Factors
  • Foxo1 protein, mouse
  • Insulin
  • Med23 protein, mouse
  • Mediator Complex
  • Cholesterol
  • RNA Polymerase II
  • Glucose