Activated platelets rescue apoptotic cells via paracrine activation of EGFR and DNA-dependent protein kinase

Cell Death Dis. 2014 Sep 11;5(9):e1410. doi: 10.1038/cddis.2014.373.

Abstract

Platelet activation is a frontline response to injury, not only essential for clot formation but also important for tissue repair. Indeed, the reparative influence of platelets has long been exploited therapeutically where application of platelet concentrates expedites wound recovery. Despite this, the mechanisms of platelet-triggered cytoprotection are poorly understood. Here, we show that activated platelets accumulate in the brain to exceptionally high levels following injury and release factors that potently protect neurons from apoptosis. Kinomic microarray and subsequent kinase inhibitor studies showed that platelet-based neuroprotection relies upon paracrine activation of the epidermal growth factor receptor (EGFR) and downstream DNA-dependent protein kinase (DNA-PK). This same anti-apoptotic cascade stimulated by activated platelets also provided chemo-resistance to several cancer cell types. Surprisingly, deep proteomic profiling of the platelet releasate failed to identify any known EGFR ligand, indicating that activated platelets release an atypical activator of the EGFR. This study is the first to formally associate platelet activation to EGFR/DNA-PK--an endogenous cytoprotective cascade.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Animals
  • Apoptosis*
  • Blood Platelets / enzymology*
  • Blood Platelets / metabolism
  • Brain / cytology
  • Brain / enzymology
  • Brain Injuries / enzymology*
  • Brain Injuries / genetics
  • Brain Injuries / physiopathology
  • Cell Line, Tumor
  • Cells, Cultured
  • DNA-Activated Protein Kinase / genetics
  • DNA-Activated Protein Kinase / metabolism*
  • ErbB Receptors / genetics
  • ErbB Receptors / metabolism*
  • Female
  • Humans
  • Male
  • Mice, Inbred C57BL
  • Middle Aged
  • Neurons / cytology*
  • Platelet Activation
  • Young Adult

Substances

  • ErbB Receptors
  • DNA-Activated Protein Kinase