Adverse hemodynamic and clinical effects of encainide in severe chronic heart failure

Ann Intern Med. 1989 Apr 1;110(7):505-9. doi: 10.7326/0003-4819-110-7-505.

Abstract

Study objective: To evaluate the hemodynamic effects of the antiarrhythmic drug, encainide, in patients with severe chronic heart failure.

Design: Unblinded, before-after study.

Setting: Referral center for patients with heart failure.

Patients: Thirty patients with severe chronic heart failure and a left ventricular ejection fraction less than 40%.

Interventions: Invasive hemodynamic measurements were done (using a balloon-tipped thermodilution catheter) before and for 3 hours after a single oral dose of 50 mg of encainide.

Measurements and main results: Ninety to one hundred and twenty minutes after its administration, encainide produced a significant deterioration in cardiac performance, as reflected by a fall in cardiac index from 2.3 to 1.8 L/min.m2 body surface (mean change 0.5 +/- 0.1; P less than 0.001), a fall in stroke work index from 26 to 18 g.m/m2 (mean change 8 +/- 2; P less than 0.001), and an increase in left ventricular filling pressure from 19 to 22 mm Hg (mean change 3 +/- 2; P less than 0.05). These deleterious hemodynamic effects were accompanied by worsening symptoms of heart failure in 8 of the 30 patients. Serum levels of encainide and its metabolites, O-desmethylencainide and 3-methoxy-O-desmethylencainide, were within the therapeutic range in most patients.

Conclusions: Encainide can cause adverse hemodynamic and clinical effects in patients with severe chronic heart failure.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Anilides / adverse effects*
  • Anilides / blood
  • Anilides / therapeutic use
  • Anti-Arrhythmia Agents / adverse effects*
  • Anti-Arrhythmia Agents / blood
  • Anti-Arrhythmia Agents / therapeutic use
  • Arrhythmias, Cardiac / complications
  • Arrhythmias, Cardiac / drug therapy
  • Dyspnea / chemically induced
  • Encainide
  • Female
  • Heart Failure / complications
  • Heart Failure / physiopathology*
  • Hemodynamics / drug effects*
  • Humans
  • Male
  • Middle Aged
  • Myocardial Contraction / drug effects
  • Stroke Volume / drug effects

Substances

  • Anilides
  • Anti-Arrhythmia Agents
  • Encainide