Effects of a new thyrotropin-releasing hormone derivative on behavioral changes after focal cerebral ischemia in rats

Stroke. 1989 Mar;20(3):362-6. doi: 10.1161/01.str.20.3.362.

Abstract

We observed the effects of a new thyrotropin-releasing hormone derivative, YM-14673 (N alpha-[[(S)-4-oxo-2-azetidinyl]carbonyl]-L-histidyl-L-prolinamide dihydrate), on behavioral changes in rats for 3 weeks after focal cerebral ischemia. Under halothane anesthesia, the left middle cerebral artery was occluded via a transretro-orbital approach. YM-14673 was administered just after the operation and once a day for 3 weeks. Neurologic deficits, including hemiplegia and abnormal posture, and disturbance of passive avoidance learning were present in solvent-treated control rats for the entire 3 weeks. YM-14673 at 0.1 or 0.3 mg/kg i.p. or 1 mg/kg p.o. significantly accelerated the recovery of neurologic deficits and ameliorated cognitive disturbance compared with the solvent-treated controls although the drug at 0.1 and 0.3 mg/kg i.p. did not influence the size of the ischemic infarct. YM-14673 mitigated the behavioral disturbances in this model of chronic focal cerebral ischemia. We also discuss the suitability of this model for the evaluation of drugs.

MeSH terms

  • Animals
  • Avoidance Learning / drug effects
  • Azetidines / pharmacology*
  • Azetines / pharmacology*
  • Behavior, Animal / drug effects*
  • Brain Ischemia / complications
  • Brain Ischemia / pathology
  • Brain Ischemia / psychology*
  • Cerebral Infarction / pathology
  • Dipeptides / pharmacology*
  • Male
  • Nervous System Diseases / etiology
  • Nervous System Diseases / physiopathology
  • Rats
  • Rats, Inbred Strains
  • Reaction Time
  • Thyrotropin-Releasing Hormone / analogs & derivatives*

Substances

  • Azetidines
  • Azetines
  • Dipeptides
  • Thyrotropin-Releasing Hormone
  • azetirelin