Reactivation of thyroglobulin gene expression in transformed thyroid cells by 5-azacytidine

Cell. 1989 Sep 22;58(6):1135-42. doi: 10.1016/0092-8674(89)90511-4.

Abstract

Transformed rat thyroid cells fail to express thyroglobulin. Cells transformed with a Kirsten murine sarcoma virus carrying a temperature-sensitive ras allele lose their transformation phenotype when shifted to the nonpermissive (39 degrees C) temperature. The thyroglobulin promoter, however, remains inactive. Similarly, transfection of these cells with a thyroglobulin promoter fused to a neomycin resistance reporter gene does not produce clones resistant to G418. Treatment of the transfected cells with the DNA demethylating agent 5-azacytidine reactivates the thyroglobulin promoter and yields stable G418-resistant clones. We show that thyroglobulin promoter activity is correlated with the presence of a thyroid-specific nuclear factor, TgTF1. TgTF1 cannot be detected in transformed cells but reappears after treatment with 5-azacytidine at 39 degrees C. Restoration of Ras activity at 33 degrees C leads to the rapid loss of TgTF1 and G418 resistance.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Azacitidine / pharmacology*
  • Base Sequence
  • Cell Line
  • Cell Nucleus / metabolism
  • Cell Transformation, Neoplastic*
  • Cloning, Molecular
  • Gene Expression Regulation / drug effects*
  • Genes / drug effects*
  • Kirsten murine sarcoma virus / genetics
  • Molecular Sequence Data
  • Oligonucleotide Probes
  • Promoter Regions, Genetic
  • Rats
  • Thyroglobulin / genetics*
  • Thyroid Gland
  • Transcription, Genetic*
  • Transfection

Substances

  • Oligonucleotide Probes
  • Thyroglobulin
  • Azacitidine