Ethanolic extracts of Tinospora cordifolia and Alstonia scholaris show antimicrobial activity towards clinical isolates of methicillin-resistant and carbapenemase-producing bacteria

Nat Prod Res. 2014;28(18):1438-45. doi: 10.1080/14786419.2014.909421. Epub 2014 Apr 22.

Abstract

The aim of this study was to determine the in vitro antimicrobial activity of crude extracts of three plants from Ayurveda tradition (Tinospora cordifolia, Alstonia scholaris, Crataeva nurvala) against reference microbial strains and clinical isolates of methicillin-resistant Staphylococcus aureus (MRSA) and carbapenemase-producing Klebsiella pneumoniae. IC50 values were obtained by micro-dilution methods meeting the requirements of the NCCLS standard. The cytotoxicity of the extracts was also investigated on a mammalian cell line. Extracts displayed a variable degree of antimicrobial activity and did not interfere with mammalian cell proliferation. T. cordifolia and A. scholaris exhibited a higher inhibitory activity against clinical isolates of MRSA and carbapenemase-producing K. pneumoniae compared with reference strains, while C. nurvala exhibited a different behaviour. An antifungal activity towards Candida albicans was observed for A. scholaris extract. Results indicate that constituents from T. cordifolia and A. scholaris may be a potential source of new therapeutic strategies for infectious diseases.

Keywords: Alstonia scholaris; Ayurveda tradition; Tinospora cordifolia; antimicrobial activity; broth micro-dilution; clinical isolates; multiple drug resistance pathogens.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alstonia / chemistry*
  • Animals
  • Anti-Infective Agents / chemistry
  • Anti-Infective Agents / isolation & purification*
  • Anti-Infective Agents / pharmacology*
  • Antifungal Agents / pharmacology
  • Bacteria / drug effects
  • Bacterial Proteins / metabolism
  • Caenorhabditis elegans / drug effects
  • Dose-Response Relationship, Drug
  • Drug Resistance, Multiple
  • Ethanol / chemistry
  • Fibroblasts / drug effects
  • Humans
  • Inhibitory Concentration 50
  • Italy
  • Klebsiella pneumoniae / drug effects
  • Medicine, Ayurvedic
  • Methicillin Resistance
  • Methicillin-Resistant Staphylococcus aureus / drug effects
  • Microbial Sensitivity Tests
  • Plant Extracts / pharmacology
  • Tinospora / chemistry*
  • beta-Lactamases / metabolism

Substances

  • Anti-Infective Agents
  • Antifungal Agents
  • Bacterial Proteins
  • Plant Extracts
  • Ethanol
  • beta-Lactamases
  • carbapenemase