Assessment of the effects of contingent histamine injections on the reinforcing effectiveness of cocaine using behavioral economic and progressive-ratio designs

Psychopharmacology (Berl). 2014 Jun;231(12):2395-403. doi: 10.1007/s00213-013-3396-y. Epub 2014 Jan 8.

Abstract

Rationale: Recent research has demonstrated that the drug, histamine, can function as a punisher of cocaine self-administration. However, little is known about how drug punishers affect the maximum reinforcing effectiveness of drugs as reinforcers.

Objective: The goal of the present study was to determine if histamine, when self-administered as a mixture with cocaine, could reduce cocaine's maximum reinforcing effectiveness using two procedures designed for measuring reinforcing effectiveness.

Methods: In the first experiment, rhesus monkeys were allowed to self-administer cocaine (0.1 mg/kg/inj) alone or as a mixture with histamine (0.012-0.05 mg/kg/inj) in a behavioral economic design. In the second experiment, monkeys were allowed to self-administer cocaine alone (0.006-0.56 mg/kg/inj) or as a mixture with histamine (0.025-0.1 mg/kg/inj) under a progressive-ratio schedule of reinforcement.

Results: In Experiment 1, histamine decreased the reinforcing effectiveness of cocaine in a dose-dependent manner as evidenced by increases in cocaine's demand elasticity with increases in histamine dose. In Experiment 2, histamine decreased cocaine's potency and effectiveness as a reinforcer in a dose-dependent manner as indicated by rightward and downward shifts, respectively, in the dose-response functions.

Conclusion: The reinforcing effectiveness of cocaine can be reduced by contingent self-administration of histamine. These results indicate that combining drug punishers with drug reinforcers reduces the maximum reinforcing effect of the drug reinforcer, which suggests a use for drug punishers as a deterrent to drug abuse (e.g., as mixtures with prescription medications with abuse potential).

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Catheters, Indwelling
  • Cocaine / pharmacology*
  • Dopamine Uptake Inhibitors / pharmacology*
  • Dose-Response Relationship, Drug
  • Economics, Behavioral
  • Histamine / pharmacology*
  • Histamine Agonists / pharmacology*
  • Macaca mulatta
  • Male
  • Reinforcement Schedule
  • Reinforcement, Psychology*
  • Self Administration

Substances

  • Dopamine Uptake Inhibitors
  • Histamine Agonists
  • Histamine
  • Cocaine