Neuregulin-1β induces embryonic stem cell cardiomyogenesis via ErbB3/ErbB2 receptors

Biochem J. 2014 Mar 1;458(2):335-41. doi: 10.1042/BJ20130818.

Abstract

NRG-1β (neuregulin-1β) serves multiple functions during embryonic heart development by signalling through ErbB family receptor tyrosine kinases (ErbB2, ErbB3 and ErbB4). Previous studies reported that NRG-1β induces cardiomyogenesis of mESCs (mouse embryonic stem cells) at the later stages of differen-tiation through ErbB4 receptor activation. In the present study we systematically examined NRG-1β induction of cardiac myocytes in mESCs and identified a novel time window, the first 48 h, for NRG-1β-based cardiomyogenesis. At this time point ErbB3, but not ErbB4, is expressed. In contrast with the later differentiation of mESCs in which NRG-1β induces cardiomyogenesis via the ErbB4 receptor, we found that knocking down ErbB3 or ErbB2 with siRNA during the early differentiation inhibited NRG-1β-induced cardiomyogenesis in mESCs. Microarray analysis of RNA expression at this early time point indicated that NRG-1β treatment in mESCs resulted in gene expression changes important to differentiation including up-regulation of components of PI3K (phosphoinositide 3-kinase), a known mediator of the NRG-1β/ErbB signalling pathway, as well as activation of CREB (cAMP-response-element-binding protein). Further study demonstrated that the NRG-1β-induced phosphorylation of CREB was required for cardiomyogenesis of mESCs. In summary, we report a previously unrecognized role for NRG-1β/ErbB3/CREB signalling at the pre-mesoderm stage for stem cell cardiac differentiation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Differentiation / genetics
  • Cell Differentiation / physiology*
  • Cell Line
  • Cyclic AMP Response Element-Binding Protein / physiology
  • Embryonic Stem Cells / physiology*
  • Gene Knockdown Techniques
  • Mice
  • Myocytes, Cardiac / physiology*
  • Nerve Tissue Proteins / physiology
  • Neuregulin-1 / physiology*
  • RNA, Small Interfering / genetics
  • Receptor, ErbB-2 / deficiency*
  • Receptor, ErbB-2 / physiology*
  • Receptor, ErbB-3 / deficiency
  • Receptor, ErbB-3 / genetics
  • Receptor, ErbB-3 / physiology*
  • Signal Transduction / physiology

Substances

  • Creb1 protein, mouse
  • Cyclic AMP Response Element-Binding Protein
  • Nerve Tissue Proteins
  • Neuregulin-1
  • RNA, Small Interfering
  • neuregulin beta
  • ERBB3 protein, human
  • Erbb2 protein, mouse
  • Receptor, ErbB-2
  • Receptor, ErbB-3