Bicarbonate-stimulated ATPase activity of bovine liver alkaline phosphatase

J Hepatol. 1985;1(2):167-78. doi: 10.1016/s0168-8278(85)80764-9.

Abstract

A commercial preparation of bovine hepatic alkaline phosphatase was found to have a Mg2+-stimulated ATPase activity. The pH optimum was 8.5, the Km for ATP was 4.2 X 10(-5) M and the Vmax was 88.3 mumol Pi . h-1 . mg-1. HCO3- had a stimulatory effect on Mg2+ -ATPase activity. Other anions had no effect or an inhibitory effect while Na+, K+ and ouabain had no effect. Purification of the commercial preparation by gel filtration and affinity chromatography yielded a fraction with alkaline phosphatase and (Mg2+ + HCO3-)ATPase activities that had been enriched respectively 27-fold and 23-fold; both activities were inhibited by levamisole (93.1% and 93.8%, respectively) and the purified fraction was found to be a single protein on sodium dodecyl sulfate polyacrylamide gel electrophoresis. These results suggest that alkaline phosphatase and (Mg2+ + HCO3-)ATPase may be properties of the same liver protein that might be involved in biliary HCO3- transport and bile secretion.

MeSH terms

  • Alkaline Phosphatase / antagonists & inhibitors
  • Alkaline Phosphatase / metabolism*
  • Animals
  • Bicarbonates / pharmacology*
  • Bile Acids and Salts / pharmacology
  • Ca(2+) Mg(2+)-ATPase / antagonists & inhibitors
  • Ca(2+) Mg(2+)-ATPase / metabolism*
  • Cattle
  • Dose-Response Relationship, Drug
  • Enzyme Activation / drug effects
  • Homoarginine / pharmacology
  • Kinetics
  • Levamisole / pharmacology
  • Liver / enzymology*
  • Ouabain / pharmacology
  • Sodium / pharmacology

Substances

  • Bicarbonates
  • Bile Acids and Salts
  • Homoarginine
  • Levamisole
  • Ouabain
  • Sodium
  • Alkaline Phosphatase
  • Ca(2+) Mg(2+)-ATPase