Stimulatory effect of ouabain on T- and L-type calcium currents in guinea pig cardiac myocytes

Am J Physiol. 1990 May;258(5 Pt 2):H1620-3. doi: 10.1152/ajpheart.1990.258.5.H1620.

Abstract

The effect of 10(-6) M ouabain on macroscopic low-threshold T-type Ca2+ and high-threshold L-type Ca2+ currents was studied by whole cell recording in isolated guinea pig ventricular myocytes superfused with K-free, Na-free media, i.e., after suppression of Na-K-ATPase activity and Na influx through the Na-Ca exchanger. Under such conditions, the amplitudes of the two currents were significantly increased by ouabain. In particular, the current occurring in the -50 to -20 mV range (T-type Ca2+) was increased two- to threefold by ouabain and suppressed by 40 microM Ni2+. Ouabain shifted by approximately 10 mV toward negative potentials the steady-state inactivation curve of the T-type Ca2+ current but not that of the L-type Ca2+ current. It is concluded that ouabain enhances not only L-type Ca2+ current but also T-type Ca2+ current possibly through different mechanisms.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cadmium / pharmacology
  • Calcium / physiology*
  • Electrophysiology
  • Guinea Pigs
  • Heart / physiology*
  • Homeostasis
  • Membrane Potentials
  • Myocardium / cytology
  • Nickel / pharmacology
  • Ouabain / pharmacology*

Substances

  • Cadmium
  • Ouabain
  • Nickel
  • Calcium