iGLuc: a luciferase-based inflammasome and protease activity reporter

Nat Methods. 2013 Feb;10(2):147-154. doi: 10.1038/nmeth.2327. Epub 2013 Jan 6.

Abstract

Measurement of protease activity in living cells or organisms remains a challenging task. We here present a transgene-encoded biosensor that reports the proteolytic activity of caspase-1 in the course of inflammasome activation and that of other proteases in a highly sensitive and specific manner. This protease reporter is based on the biological activity of a pro-interleukin (IL)-1β-Gaussia luciferase (iGLuc) fusion construct, in which pro-IL-1β-dependent formation of protein aggregates renders GLuc enzyme inactive. Cleavage leads to monomerization of this biosensor protein, resulting in a strong gain in luciferase activity. Exchange of the canonical caspase-1 cleavage site in this reporter construct allows the generation of protease biosensors with additional specificities. The high sensitivity, signal-to-background ratio and specificity of the iGLuc system renders it a useful tool to study proteolytic events in mouse and human cells at high throughput and to monitor protease activity in mice in vivo.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biosensing Techniques / methods*
  • Caspase 1 / metabolism
  • Cell Line
  • Enzyme Activation
  • Humans
  • Inflammasomes / metabolism*
  • Interleukin-1beta / metabolism*
  • Luciferases / metabolism*
  • Mice
  • Transfection

Substances

  • Inflammasomes
  • Interleukin-1beta
  • Luciferases
  • Caspase 1