The effects of Di-(2-ethylhexyl)-phthalate exposure on fertilization and embryonic development in vitro and testicular genomic mutation in vivo

PLoS One. 2012;7(11):e50465. doi: 10.1371/journal.pone.0050465. Epub 2012 Nov 30.

Abstract

The present study was undertaken to determine the reproductive hazards of Di-(2-ethylhexyl)-phthalate (DEHP) on mouse spermatozoa and embryos in vitro and genomic changes in vivo. Direct low-level DEHP exposure (1 μg/ml) on spermatozoa and embryos was investigated by in vitro fertilization (IVF) process, culture of preimplanted embryos in DEHP-supplemented medium and embryo transfer to achieve full term development. Big Blue® transgenic mouse model was employed to evaluate the mutagenesis of testicular genome with in vivo exposure concentration of DEHP (500 mg/kg/day). Generally, DEHP-treated spermatozoa (1 μg/ml, 30 min) presented reduced fertilization ability (P<0.05) and the resultant embryos had decreased developmental potential compared to DMSO controls (P<0.05). Meanwhile, the transferred 2-cell stage embryos derived from treated spermatozoa also exhibited decreased birth rate than that of control (P<0.05). When fertilized oocytes or 2-cell stage embryos were recovered by in vivo fertilization (without treatment) and then exposed to DEHP, the subsequent development proceed to blastocysts was different, fertilized oocytes were significantly affected (P<0.05) whereas developmental progression of 2-cell stage embryos was similar to controls (P>0.05). Testes of the Big Blue® transgenic mice treated with DEHP for 4 weeks indicated an approximately 3-fold increase in genomic DNA mutation frequency compared with controls (P<0.05). These findings unveiled the hazardous effects of direct low-level exposure of DEHP on spermatozoa's fertilization ability as well as embryonic development, and proved that in vivo DEHP exposure posed mutagenic risks in the reproductive organ - at least in testes, are of great concern to human male reproductive health.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blastocyst / drug effects*
  • Diethylhexyl Phthalate / pharmacology*
  • Embryo Transfer
  • Embryo, Mammalian
  • Embryonic Development / drug effects*
  • Female
  • Fertilization / drug effects*
  • Fertilization in Vitro
  • Humans
  • Male
  • Mice
  • Mice, Transgenic
  • Mutation
  • Oocytes / drug effects*
  • Plasticizers / pharmacology*
  • Pregnancy
  • Reproduction / drug effects
  • Reproduction / physiology
  • Sperm Motility / drug effects
  • Spermatozoa / drug effects*
  • Testis / cytology
  • Testis / drug effects*

Substances

  • Plasticizers
  • Diethylhexyl Phthalate

Grants and funding

The research was supported by the grants as follows: the Major State Basic Research Development Program of China (973 Program, 2009CB941700), the grants from National Natural Science Foundation of China (81270744), Three National Comprehensive Programs of Reproductive Health and Family Planning (C1-93) and Shanghai Leading Academic Discipline Project (S30201). The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.