Inefficient vaginal transmission of tenofovir-resistant HIV-1

J Virol. 2013 Jan;87(2):1274-7. doi: 10.1128/JVI.01777-12. Epub 2012 Oct 31.

Abstract

Transmission of drug-resistant HIV has been postulated to be a threat to current first-line antiretroviral therapy (ART) regimens and the efficacy of several antiretroviral-based preexposure prophylaxis (PrEP) strategies being tested. Here we evaluated the effect of the common tenofovir (TFV) resistance mutation K65R on vaginal HIV transmission. Our results demonstrate that despite no overt loss of overall replication competence in vivo, this mutation results in significantly reduced mucosal transmission. When transmitted, the mutant virus eventually reverted to the wild type in 2 of 3 animals examined.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / pharmacology
  • Animals
  • Anti-HIV Agents / pharmacology*
  • Disease Models, Animal
  • Drug Resistance, Viral*
  • Female
  • Genotype
  • HIV Infections / transmission*
  • HIV Infections / virology*
  • HIV-1 / classification
  • HIV-1 / drug effects*
  • HIV-1 / genetics
  • Humans
  • Mice
  • Mucous Membrane / virology
  • Mutation, Missense*
  • Organophosphonates / pharmacology*
  • Suppression, Genetic
  • Tenofovir
  • Vagina / virology

Substances

  • Anti-HIV Agents
  • Organophosphonates
  • Tenofovir
  • Adenine