Protective effects of nebivolol against anthracycline-induced cardiomyopathy: a randomized control study

Int J Cardiol. 2013 Sep 1;167(5):2306-10. doi: 10.1016/j.ijcard.2012.06.023. Epub 2012 Jun 22.

Abstract

Background: We aimed to evaluate the effect of prophylactic nebivolol use on prevention of antracycline-induced cardiotoxicity in breast cancer patients.

Methods: In this small, prospective, double-blind study, we randomly assigned 45 consecutive patients with breast cancer and planned chemotheraphy to receive nebivolol 5mg daily (n=27) or placebo (n=18). Echocardiographic measurements and N-terminal pro-brain natriuretic peptide (NT-pro-BNP) levels were obtained at baseline and at 6-month of chemotherapy.

Results: Both studied groups had comparable echocardiographic variables and NT-pro-BNP levels at baseline. At 6-month, the left ventricular (LV) end-systolic and end-diastolic diameters increased in the placebo group (LVESD: 29.7 ± 3.4 to 33.4 ± 4.5mm; LVEDD: 47.2 ± 3.8 to 52.0 ± 4.6mm, p=0.01 for both) but remained unchanged in the nebivolol group (LVESD: 30.4 ± 3.5 to 31.0 ± 3.6mm, p=0.20; LVEDD: 47.0 ± 4.4 to 47.1 ± 4.0mm, p=0.93). The placebo group also had lower LVEF than the nebivolol group (57.5 ± 5.6% vs. 63.8 ± 3.9%, p=0.01) at 6-month. NT-pro-BNP level remained static in the nebivolol group (147 ± 57 to 152 ± 69 pmol/l, p=0.77) while it increased in the placebo group (144 ± 66 to 204 ± 73 pmol/l, p=0.01).

Conclusions: Prophylactic use of nebivolol treatment may protect the myocardium against antracycline-induced cardiotoxicity in breast cancer patients.

Keywords: Anthracycline; Cardiomyopathy; Nebivolol.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Adult
  • Anthracyclines / adverse effects*
  • Antineoplastic Agents / adverse effects
  • Benzopyrans / administration & dosage*
  • Cardiomyopathies / chemically induced*
  • Cardiomyopathies / diagnostic imaging
  • Cardiomyopathies / prevention & control*
  • Cardiotonic Agents / administration & dosage*
  • Double-Blind Method
  • Ethanolamines / administration & dosage*
  • Female
  • Humans
  • Middle Aged
  • Nebivolol
  • Prospective Studies
  • Ultrasonography

Substances

  • Anthracyclines
  • Antineoplastic Agents
  • Benzopyrans
  • Cardiotonic Agents
  • Ethanolamines
  • Nebivolol