Histamine receptor assays

Curr Protoc Pharmacol. 2001 Nov:Chapter 4:Unit4.17. doi: 10.1002/0471141755.ph0417s14.

Abstract

This unit describes three standard in vitro bioassays for studying histamine H₁, H₂ and H₃ receptors in isolated intact tissues removed from the guinea pig. Both the H₁ and H₃ receptor assays are based on preparations of the ileum, whereas the spontaneously beating right atrium assay is used for the H₂-receptor.This unit describes three standard in vitro bioassays for studying histamine H₁, H₂ and H₃ receptors in isolated intact tissue.

MeSH terms

  • Animals
  • Guinea Pigs
  • Histamine Agonists / metabolism
  • Histamine Antagonists / metabolism
  • Ileum / metabolism*
  • In Vitro Techniques
  • Male
  • Radioligand Assay / methods*
  • Receptors, Histamine / metabolism*

Substances

  • Histamine Agonists
  • Histamine Antagonists
  • Receptors, Histamine